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Haem-activated promiscuous targeting of artemisinin in Plasmodium falciparum

$ 19.99

4.6 (113) In stock

PDF] Rapid kill of malaria parasites by artemisinin and semi-synthetic endoperoxides involves ROS-dependent depolarization of the membrane potential

Advances in the research on the targets of anti-malaria actions of artemisinin. - Abstract - Europe PMC

Dual-pharmacophore artezomibs hijack the Plasmodium ubiquitin-proteasome system to kill malaria parasites while overcoming drug resistance - ScienceDirect

Artemisinin acts by inhibiting Plasmodium falciparum Ddi1, a retropepsin, resulting into the accumulation of ubiquitinated proteins

Plasmodium falciparum: multifaceted resistance to artemisinins, Malaria Journal

Artemisinin targets are involved in multiple biological processes

Decreased K13 Abundance Reduces Hemoglobin Catabolism and Proteotoxic Stress, Underpinning Artemisinin Resistance - ScienceDirect

Artemisinin-resistant K13 mutations rewire Plasmodium falciparum's intra-erythrocytic metabolic program to enhance survival

Artemisinin activation in P. falciparum relies on two distinct haem

Artemisinin Action and Resistance in Plasmodium falciparum. - Abstract - Europe PMC

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